http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-104892485-B
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-60 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-42 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-60 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-42 |
| filingDate | 2015-06-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2018-03-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2018-03-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CN-104892485-B |
| titleOfInvention | 2 perfluoroalkyl indole derivativeses and its synthetic method |
| abstract | The present invention relates to a kind of 2 perfluoroalkyl indole derivativeses and its synthetic method, the structure of the compound to be： Wherein R F For C 1 —C 3 Perfluoroalkyl.The inventive method is used as raw material using the anil and the perfluoroalkyl acetylenic acid ester of synthesis gimmick maturation being easy to get, under certain condition, the indole derivatives containing perfluoroalkyl by Michael additions and C H activation synthesis, compared with traditional approach synthesizes similar product, this method is initiation material using aniline and acetylenic, can expand the selectivity of substrate significantly；And this method is skimmed traditional oxidant in oxidizing process, by the use of oxygen as oxidant, green and the theory of sustainability chemistry are embodied.Regioselectivity is high, and yield is good.Therefore this method is to synthesize effective new method of 2 perfluoroalkyl indole derivativeses. |
| priorityDate | 2015-06-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 70.