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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K51-00
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K1-13
filingDate 2013-11-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-10-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2018-10-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-104854126-B
titleOfInvention polypeptide and imaging method
abstract The present invention provides a kind of peptide, and the peptide can be used as the image probe of GLP 1R.In a mode, the polypeptide indicated with formula (3) is provided.Xaa 1 Leu Ser Lys Gln Met Glu Glu Glu Ala Val Arg Leu Phe Ile Glu Trp Leu Lys Asn Gly Gly Pro Ser Ser Gly Ala Pro Pro Pro Ser (3) (sequence number 3) are in formula (3), Xaa 1 It is the aspartic acid that Y X ' bases are incorporated in α amino, X ' includes chelating portion and the radioactive metal nucleic being chelated in the chelating portion, the chelating portion is diethylene triamine base pentaacetic acid dianhydride (DTPA) or 1,4,7 triazododecane N, N ', N " triacetic acid (NOTA), Y are to include from by CH 2 ‑(C 6 H 4 ), NH C (=S) and NH (CH 2 ) 5 The connexon of the base selected in the group that C (=O) and combination thereof are constituted.
priorityDate 2012-11-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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