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filingDate 2013-06-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2016-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-104684922-B
titleOfInvention (E) prodrug derivant of-N-methyl-N-((3-methyl benzofuran-2-base) methyl)-3-(7-oxo-5,6,7,8-tetrahydrochysene-1,8-naphthyridines-3-base) acrylamide
abstract A part of the present invention relates to (E) N methyl N, and (derivant of (3 methyl 1,8 naphthyridines 3 base) acrylamide compound, it has noticeable dissolubility, solid-state stability and bioavailability characteristics.Find that described compound is by effective inhibitor that effectively suppression FabL hi addition is bacterial fatty acid metabolic, it was demonstrated that some compound is stable for gamma-radiation sterilization treatment, is therefore very suitable for preparing the sterile preparation being infected the disease caused for treatment by antibacterial.
priorityDate 2012-06-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 429.