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filingDate 2013-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3ff3e8d2f3bf7fd2fa0495ec6987e84d
publicationDate 2015-03-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-104415026-A
titleOfInvention Application of deuterated fumaric acid-enriched derivative in treatment of multiple sclerosis
abstract The invention relates to application of a deuterated fumaric acid-enriched derivative in preparation of medicaments for treating or preventing multiple sclerosis. The deuterated fumaric acid-enriched derivative is selected from the following components: 2,3-dideuterium- or 2-deuterium- or 3-deuterium-dialkyl fumarate, 2,3-dideuterium- or 2-deuterium- or 3-deuterium-hyrogen monoalkyl fumarate, 2,3-dideuterium- or 2-deuterium- or 3-deuterium-salt monoalkyl fumarate, 2,3-dideuterium- or 2-deuterium- or 3-deuterium-monoamide fumarate, 2,3-dideuterium- or 2-deuterium- or 3-deuterium-salt monoamide fumarate, 2,3-dideuterium- or 2-deuterium- or 3-deuterium-diamide fumarate and 2,3-dideuterium- or 2-deuterium- or 3-deuterium-monoalkyl monoamide fumarate as well as the mixture of the compounds. The application is found based on the fact that cellular pathways of Nrf2 in cells can be activated by the deuterated fumaric acid derivative.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2023045377-A1
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type http://data.epo.org/linked-data/def/patent/Publication

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