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filingDate 2013-03-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-04-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2018-04-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-104363924-B
titleOfInvention Control for delivering 1 inhibitor of HIF discharges composite
abstract The Controlled release formulation amount composite for being used for delivering one or more 1 inhibitor of HIF is provided.The control release composite contains one or more and is incorporated into or is scattered in 1 inhibitor of HIF in polymer mediator.In some cases, one or more 1 inhibitor of HIF are dispersed in or are packaged in polymer substrate.In a preferred embodiment, one or more described 1 inhibitor of HIF are covalently bonded in polymer, form polymeric medicine conjugate.Polymer mediator can form the implant for administering, particulate, nano-particle or its combination.Control release 1 composites of HIF provide long-term treatment benefit by discharging one or more 1 inhibitor of HIF and/or 1 inhibitor conjugates of HIF of low content within an elongated segment period, while reduce side effect.Controlled release formulation amount composite for delivering one or more 1 inhibitor of HIF can be used for treating or preventing disease or illness related with vascularization in patient, including cancer, obesity and eye disease, such as moist AMD.
priorityDate 2012-03-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 469.