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filingDate 2014-09-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_88461899baf780c33abf9655e15f0ecc
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publicationDate 2015-01-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-104311471-A
titleOfInvention A kind of industrial preparation method of improved mitiglinide calcium
abstract The present invention is an improved preparation method of mitiglinide calcium (I), which is characterized in that: the preparation method successively comprises step 1: preparation of 2-benzylidene succinic acid; step 2: (S)-2-benzyl Preparation of phenylsuccinic acid; Step 3: 2-(S)-Benzyl-4-oxo-(cis-perhydroisoindol-2-yl)butanoic acid; Step 4: Preparation of mitiglinide calcium . The invention provides an economical and practical method for industrialized preparation of mitiglinide calcium with simple operation, short reaction period and high yield.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-107963989-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-109081805-A
priorityDate 2014-09-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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