Predicate |
Object |
assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_bf22b6e9a2c2da5ae7b3c452f577492b |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-44 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-44 |
filingDate |
2014-09-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_88461899baf780c33abf9655e15f0ecc http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5ee38f7f698f3754c7cbe8174da4ef9e http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c310d8b74691b63e43398735722244e5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1425880598458aebf30e3f99892ecbaa http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6545dedc18dc89bd740bd3066a3ea924 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b94841054cd4c0a1e3d5fca35d3e3566 |
publicationDate |
2015-01-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
CN-104311471-A |
titleOfInvention |
A kind of industrial preparation method of improved mitiglinide calcium |
abstract |
The present invention is an improved preparation method of mitiglinide calcium (I), which is characterized in that: the preparation method successively comprises step 1: preparation of 2-benzylidene succinic acid; step 2: (S)-2-benzyl Preparation of phenylsuccinic acid; Step 3: 2-(S)-Benzyl-4-oxo-(cis-perhydroisoindol-2-yl)butanoic acid; Step 4: Preparation of mitiglinide calcium . The invention provides an economical and practical method for industrialized preparation of mitiglinide calcium with simple operation, short reaction period and high yield. |
isCitedBy |
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-107963989-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-109081805-A |
priorityDate |
2014-09-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |