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filingDate 2012-12-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2014-10-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-104114183-A
titleOfInvention CTP-based insulin analogs for the treatment of diabetes
abstract Insulin analogues comprising non-native glycosylation site sequences having high potency and specificity for the insulin receptor are provided. In one embodiment, a peptide sequence greater than 18 amino acids is used as a linking moiety linking human insulin A and B chains or analogs or derivatives thereof to provide a high potency single chain insulin analog. In one embodiment, the linking moiety comprises one or more glycosylation sites. Prodrug and conjugate derivatives of the insulin analogs are also disclosed.
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