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filingDate 2013-07-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2c4bc3da8a9cb145dd4fe5bd1b03b0c7
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publicationDate 2015-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-103360312-B
titleOfInvention Geldanamycin derivative and its application
abstract The invention discloses a geldanamycin derivative is a 17-mono-substituted or 17,19-disubstituted geldanamycin derivative, structural general formula of which is as shown in the formula (I). It is confirmed through experiments that the geldanamycin derivative maintains or increases its original antineoplastic activity and obviously reduces its hepatotoxicity, thus laying a foundation for research and development of an antitumor drug with the geldanamycin derivative used as a lead compound.
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