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Predicate Object
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D223-22
filingDate 2013-02-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-08-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2015-08-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-103288736-B
titleOfInvention A kind of preparation method of eslicarbazepine intermediate
abstract The invention discloses a kind of preparation method of eslicarbazepine intermediate, it is with 5H-dibenzo [B, F] azepine-10 (11H)-one (compound III) is raw material, react with phosgene, trichloromethylchloroformate, triphosgene, chloro-formic ester compounds or chloroformyl sulphinyl chlorine, obtain Compound II per; Compound II per carries out ammonolysis reaction and obtains final product under the existence of ammonia; Present invention process route is shorter, and low in raw material price is simple and quick, and cost is lower, is applicable to suitability for industrialized production.
priorityDate 2013-02-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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