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classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-18
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-519
filingDate 2011-09-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2016-02-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-02-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-102993200-B
titleOfInvention Paliperidone amino-acid ester and preparation method thereof
abstract The present invention discloses and is a kind ofly used for the treatment of the compound Paliperidone amino-acid ester of mental disorder or the preparation method of its pharmaceutical salts, and its structural formula is (I).This compounds also can be able to be both racemic mixture for optically active isomer.Such Paliperidone amino-acid ester can metabolic conversion be the paliperidone (II) with pharmacologically active through taking in after in body in vivo, as the Antagonists exert drug effect of transmitter substance, and the relevant mental disorder such as treatment schizophrenia.
priorityDate 2011-09-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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