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filingDate 2011-05-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2016-10-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-10-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-102784096-B
titleOfInvention A kind of Asiatic acid self-microemulsifyindrug drug delivery system and preparation method thereof
abstract The invention discloses a kind of Asiatic acid self-microemulsifyindrug drug delivery system (AA SMEDDS) and preparation method thereof.Comprising: 0.5%~5% asiatic acid, oil phase 10% 50%, emulsifying agent 30% 75% and co-emulsifier 0% 30%, percentage ratio is mass percent.Preparation method comprises the following steps: weigh appropriate asiatic acid, adds co-emulsifier and the emulsifying agent of recipe quantity, makes it dissolve 25~45 DEG C of stirrings, then according to recipe quantity adds oil phase and other adjuvants, stirs and get final product.The asiatic acid self-emulsifying microemulsion oral preparation composition of the present invention, after oral chance body fluid, spontaneous emulsification becomes the emulsion droplet of its below particle diameter 100nm.Preparation is simple, and medicine stability is good, and bioavailability is high.
priorityDate 2011-05-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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