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publicationDate 2012-10-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-102713618-A
titleOfInvention Protein Kinase Complexes and Inhibitors
abstract The present invention relates to a protein complex comprising a protein kinase comprising a cysteine residue located at the ATP binding site and an inhibitor covalently and irreversibly binds to said cysteine residue, so that the activity of said protein kinase is irreversibly inhibited. The invention also relates to compounds for the irreversible inhibition of protein kinases.
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