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filingDate 2009-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2014-08-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_419f28913db0c4b653ec69a5c26e84df
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_601c19976e89d0375a62f5cbdd65c1c3
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publicationDate 2014-08-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-102186844-B
titleOfInvention Radiolabelled inhibitors of the glycine 1 transporter
abstract The present invention relates to novel radiolabelled inhibitors of general formula (I) for the Glycine 1 transporter (GlyT1), useful for the labelling and diagnostic imaging of the glycine 1 transporter functionality. Wherein R1 is isopropoxy or 2,2,2-trifluoro-1-methyl-ethoxy; and R2 is a radiolabelled group CH3, wherein the radionuclide is 3H or 11C. It has been found that the radiolabelled compounds of formula (I) may be used as PET (Positron Emission Tomography) radiotracer for the labelling and diagnostic molecular imaging of the glycine 1 transporter functionality.
priorityDate 2008-11-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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