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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D213-73
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filingDate 2006-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9783c9194d6368f9912c36d76a78689f
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_398237cc083b05bdffe0e42e04d6a3f4
publicationDate 2008-08-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-101243069-A
titleOfInvention Thrombin inhibiting 2-oxo-1,2,5,6-tetrahydropyridine derivatives
abstract There is provided a compound of formula (I) wherein R<1>, R<2a>, R<2b>, R<3a>, R<3b>, R<4>, R<5a>, R<5b>, R<6> to R<8>, A and G have meanings given in the description, which compounds are useful as, or are useful as prodrugs of, competitive inhibitors of trypsin-like proteases, such as thrombin, and thus, in particular, in the treatment of conditions where inhibition of thrombin is beneficial (e.g. conditions, such as thrombo-embolisms, where inhibition of thrombin is required or desired, and/or conditions where anticoagulant therapy is indicated).
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-113698386-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-113698386-B
priorityDate 2005-06-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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