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publicationDate 2019-10-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CL-2019001514-A1
titleOfInvention Process for the preparation of (s) -5- (r2) -n- (2-hydroxy-2-methylpropyl) -4- (2-methylpyrrolidine-1-carbonyl) thiazole-2-carboxamide (divisional of application 436 -2018)
abstract A method for preparing a (S) -5- (R 2) -N- (2-hydroxy-2-methylpropyl) -4- (2-methylpyrrolidine-1-carbonyl) thiazole-2-carboxamide comprising the reaction step (S ) -N- (2-hydroxy-2-methylpropyl) -4- (2-methylpyrrolidine-1-carbonyl) thiazole-2-carboxamjda, R 2 -Br, K2CO3, Pivalic acid, Pd2 (dba) 3.CHCI3 and cataCXium A, where R2 is selected from the group.
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