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filingDate 2011-11-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c881b392d98e3f93f8e8a7d624e60530
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publicationDate 2012-04-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CL-2011002837-A1
titleOfInvention Compounds derived from 1,2,4-triazolo [4,3-a] pyridine, positive allosteric modulators of mglur2 receptors; pharmaceutical composition; process to prepare it; and its use in the treatment or prevention of a central nervous system disorder such as anxiety, schizophrenia and migraine, among others.
abstract COMPOUNDS DERIVED FROM TRIAZOLO (4, 3-A) PYRIDINE OF FORMULA (I) ARE DESCRIBED. WHERE ALL THE RADICALS ARE AS DEFINED IN THE CLAIMS. THE COMPOUNDS IN ACCORDANCE WITH THE INVENTION ARE POSITIVE ALLOSTERIC MODULATORS OF THE METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 2 ("MGLUR2"), WHICH ARE USEFUL FOR THE TREATMENT OR PREVENTION OF NEUROLOGICAL DISORDERS AND DISEASES OF GLUTAMATE DISEASES IN DISEASED GLUTAMETTE AND SIQUIATRICOS IN THE CONDITION OF GLUTAMMATE SIQUIATRIC MGLUR2 SUBTYPE OF METABOTROPIC RECEPTORS IS INVOLVED. THE INVENTION FURTHER REFERS TO PHARMACEUTICAL COMPOSITIONS INCLUDING SUCH TYPE OF COMPOUNDS, TO PROCESSES FOR PREPARING SUCH COMPOUNDS AND COMPOSITIONS, AND TO THE USE OF SUCH TYPE OF COMPOUNDS FOR THE PREVENTION OR TREATMENT OF INVOLVED NEUROLOGICAL DISORDERS AND MUSCED NEUROLOGICAL AND SIQUAD . <br />
priorityDate 2009-05-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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