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filingDate 1967-05-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1973-09-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CH-539436-A
titleOfInvention Process for the dissolution of drugs containing basic reacting nitrogen atoms
abstract Preparation of soluble basic medicaments having one or more basic nitrogen atoms in their structure, esp. basic xanthine derivatives e.g theophylline and theobromines T - Alk - NH - CHR1CHR2R3 T=dialkylxanthinyl- Alk=C2-6 alkylene R1=H or lower alkyl- R2=H or OH R3=phenyl or hydroxyphenyl-. by reacting the basic medicament with an aryl-sulphonic acid R'1 and R'2 = same of different H-, phenyl-, C1-5 alkylphenyl-, alkyl which may form a ring opt. through O or N esp. benzene sulphonic acid, p-toluene sulphonic acid, D,L-camphorsulphonic acid, cyclohexylamidosulphuric acid. Preparation of soluble basic injections and aerosols.
priorityDate 1966-06-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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