abstract |
(A) Benzodiazepine derivs. of the general formula (I):- R1,R5 = H, alkyl, alkenyl, alkynyl, -CnH2n-halogen(P), -CnH2nNR7R8(Q); at least one of R1 and R5 must be P or Q. R2 = H, alkyl R3 = H, halogen, CF3, NO2 R4 = H, halogen, CF3, NO2, alkyl-S R6 = H, or with R5, a C-N bond R7,R8 = alkyl or NR7R8 = monoheterocycle (may contain 1 more O or N atom) n = 2-7 Anticonvulsants, analgesics, sedatives and muscle relaxants. |