http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-2931592-A1

Outgoing Links

Predicate Object
assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_2dfde99b696148d6c84b5dfb50916f23
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-2054
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-08
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-0095
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-10
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K45-06
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-40
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-0056
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-2009
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-2013
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-2018
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-2027
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-2031
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-40
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-401
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-20
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-28
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-48
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-20
filingDate 2014-12-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6e1bcfa1a8a8bf11de3a9ebe7bd8afba
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3bd8315d30fd0b6bdefc639ecb1ee75b
publicationDate 2015-06-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2931592-A1
titleOfInvention Oral formulations of pyrrolidine derivatives
abstract In the management of preterm labor and premature birth, there is a need for an oral formulation which is convenient to administer, which is suitable for providing a fast onset of action and which provides a good bioavailability of a compound being an OT-R antagonist.Accordingly, the present invention relates to a dispersible tablet comprising a compound of formula (3Z,5S)-5-(hy droxymethy 1)- 1- [(2' -methy 1- 1, 1 '-bipheny 1-4-y 1)carbonyllpy rroli di n-3 -one-O-methyloxime and at least one or more pharmaceutically acceptable excipients. The invention also provides said dispersible tablet, for use in the treatment and/or prevention of disorders selected from the group comprising preterm labor, premature birth, embryo implantation failure due to uterine contractions, dysmenorrhea, premature ejaculation, sexual dysfunction, endometriosis, infertility, benign prostatic hyperplasia, neuro-psychiatric disorders, autism, social behavior disorders, psycho-social stress, and/or cardiovascular disorders. Also provided is a process for the preparation of said dispersible tablet characterized by a step of wet granulation. The invention further provides a kit comprising said dispersible tablet, and information for use thereof.
priorityDate 2013-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

Incoming Links

Predicate Subject
isDiscussedBy http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2083
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448718630
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453694953
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448783041
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID339493
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504952
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10236
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534805
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID20722760
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID439302
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID62726
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID552
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2662
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506158
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25203916
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1548887
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280888
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448316871
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453678473
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5311010
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11397538
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP42672
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10239
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419538410
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411574743
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453808416
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24414
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452135712
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415853316
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5TJ03
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP30202
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14941
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419508054
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68986
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID62223
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419549665
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68985
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4813803
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419762300
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448178750
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452788844
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID352922
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID442979
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451577746
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423352616
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5234
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID538439
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453467280
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454570538
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419489866
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09569
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5090
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506282
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13836
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID61680
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16703273
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280728
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5281
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24456
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449282311
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5102882
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15324
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID417430547
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21252321
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8JN66
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9IIH4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ83906
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4485
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID174
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11556
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419557062
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ84177
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10176082
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID233208
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO40958
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502692
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415731092
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID114690
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448670727
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5460770
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP03253
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419490523
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100152272
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP03252
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID517055
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450984220
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422140505
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID168533
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14792
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416053122
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID54140
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25504
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9782
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452983531
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453754419
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559553
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24497
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449454525
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5780
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419591227
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24832091
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154496863
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451363760
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID644077
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492800
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419527835
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6912
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506910
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4495
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134688829
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733267
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID702
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448277656
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534410
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24221
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO71150
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419579320
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412667134
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID18429
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24261
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO71070
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID155
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10449793
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11029
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419563633
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421304351
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281606
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID151263
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419577855
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453030527
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426323564
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID87540
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507320
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24682
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID339493
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409282571
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419555446
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453998568
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396101
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6251
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23668838
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24832095
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23665634
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450364447
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5793
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID430991
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5020
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419555450
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID699129
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID84571
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426260389
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3033836
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9WF19
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426260513
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10415276
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18351450
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5743
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457707758
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426260387
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10112
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25107
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6328154
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449760797
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419490943
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502508
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6917
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419546934
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24846132
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9QM72
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419491805
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6106
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11825
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448546691
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07885
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452927767
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3454
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11826
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID92024010
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2759815
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID82170
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11177
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419514741
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25645
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID33572
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3084116
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433322677
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4510
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID464113
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID87540
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433323226
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9831860
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419553385
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5460341
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID114548
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID521874
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3423265
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419524794
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19151
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419546958
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID51064083
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421281770
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504692
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ96629
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11998
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419585166
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448380735
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19119
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID551
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID571591
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5403
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP87563
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11464
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8221
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68984
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID352920
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5360545
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10381
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449950617
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID38288
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419527161
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5143
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426384952
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24699
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559505

Total number of triples: 252.