http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-2770766-A1

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filingDate 2010-08-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4818fb9aa85f57c6aea1d0bac077ab09
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4f6a778fc1f077f185de01b4b31eb6b3
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_257c225d63e6dc9baa2dd4b9cb32d3f6
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b038d730a9e633a4d2f7de0dd9fdca9a
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3e84f1e4485d3d1e2cf42af7b5987ada
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b92f553aaf08461a651508b32ad96df5
publicationDate 2011-02-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2770766-A1
titleOfInvention Disubstituted [4-(5-aminomethyl-phenyl)-piperidin-1-yl]-1h-indol-3-yl]-methanones
abstract The present invention extends to the compound of formula I: or a prodrug, pharmaceutically acceptable salt, or solvate of said compound. Furthermore, the present invention is directed to a pharmaceutical composition comprising a pharmaceutically effective amount of the compound of formula I, and a pharmaceutically acceptable carrier. Furthermore, the present invention is directed to the use of a compound of formula I as an inhibitor of tryptase, comprising introducing the compound into a composition comprising tryptase. In addition, the present invention is directed to the use of a compound of formula I for treating a patient suffering from, or subject to, a physiological condition in need of amelioration of an inhibitor of tryptase comprising administering to the patient a therapeutically effective amount of the compound of Claim 1. The present invention is directed also to the preparation of a compound of formula I.
priorityDate 2009-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 528.