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filingDate 2009-12-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2013-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2747777-C
titleOfInvention A method for preparing entecavir and intermediates thereof
abstract Entecavir is a nucleoside analog and a useful antiviral agent. The present invention relates to methods for preparing entecavir of formula (1) and to intermediates used in such methods: (see formula 1) The methods of preparation are characterized by the steps of synthesizing a chiral ketone and using a .alpha.-hydroxy ketone as an intermediate.
priorityDate 2008-12-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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