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filingDate 2007-06-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6ef8958db5c681ad246c7160f2d1edff
publicationDate 2008-01-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2654394-A1
titleOfInvention Tricyclic heteroaryl compounds as pde10 inhibitors
abstract The invention pertains to tricyclic heteroaryl compounds of formula (I) that serve as effective phosphodiesterase (PDE) inhibitors. The invention also relates to compounds which are selective inhibitors of PDElO. The invention further relates to pharmaceutical compositions comprising such compounds; and the use of such compounds in methods for treating certain central nervous system (CNS) or other disorders. The invention relates also to methods for treating neurodegenerative and psychiatric disorders, for example psychosis and disorders comprising deficient cognition as a symptom.
priorityDate 2006-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A0U1RPR8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WQ35
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ25263
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423192479
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Z3Q0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID565259
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9VEU5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP43524
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID297
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9VEU6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5SDA5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A1C5G2V9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410023599
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP97490
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP30804
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40136
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423192439
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5460179
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70913
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423192478
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID524624
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559043
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23466
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419556970
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ96PN6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO88444
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID644017
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID402
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428120378
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP33402
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ57692
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ02108
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410554345
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ04400
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1Q257
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100124505
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559578
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID564465
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451750347
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394811
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GYQ4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559581
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457169682
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4ZHR9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID424116
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4ZHS0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP98999
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5288393
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP16066
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420239903
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ19187
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID456921
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8C0T9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ26721
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403652
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ76L33
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69185169
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ19768
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ26896
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19687
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ76L34
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20595
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415764221
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ52915
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457493614
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27580

Total number of triples: 381.