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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D457-06
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D457-06
filingDate 2006-03-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f58531252880ca2f43782330fb0dbe1e
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9852b38e0701a60c3adab9d563a9c69d
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a966c38299b8263d06310405c01abe22
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fd6a39244c89a70e04bed923fb22c6ab
publicationDate 2006-09-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2602898-A1
titleOfInvention Preparation of cabergoline
abstract A method of preparing cabergoline Form I, comprising forming a solvate including cabergoline and a p-disubstituted benzene of formula (A) or 1,3,5-trimethylbenzene and obtaining cabergoline Form I from the solvate. Another aspect of the present invention provides a method for preparing cabergoline Form I comprising dissolving cabergoline in p-disubstituted benzene or 1,3,5-trimethylbenzene and recovering the cabergoline Form I polymorph, suitably by direct crystallization of Form I or by recovery of a solvate which can be converted to Form I. Another aspect of the present invention provides a novel cabergoline polymorph designated cabergoline Form FB and a method of preparing said polymorph by dissolving or forming a solvate of cabergoline in fluorobenzene and recovering cabergoline Form FB.
priorityDate 2005-03-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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