http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-2582985-A1

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filingDate 2005-10-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_cde783c526fac3f40becce44452acac8
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f4ffd97b6b0d1886d7e542c83683c3b7
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publicationDate 2006-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2582985-A1
titleOfInvention Disubstituted pyrazolobenzodiazepines useful as inhibitors for cdk2 and angiogesis, and for the treatment of breast, colon, lung and prostate cancer
abstract The present invention provides compounds of the formula (I) wherein R1, R2, R3 and R4 are described herein. The invention also provides syntheses for preparation of such compounds and pharmaceutical compositions containing them. The invention further provides methods for inhibiting kinases, in particular CDK2, for inhibiting angiogenesis, and for treating cancers, in particular breast, colon, prostate, and lung cancer.
priorityDate 2004-10-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 488.