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filingDate 2004-08-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2010-09-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8cd6d70fdcb396b7808e3b07ad583c55
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_55fca8a98bb9ec5b6d311449448c9672
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publicationDate 2010-09-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2536929-C
titleOfInvention 2-substituted benzimidazole piperidines analogs as selective melanin concentrating hormone receptor antagonists for the treatment of obesity and related disorders
abstract The present invention discloses compounds of formula (I); wherein Ar, Y, m, n, R1 and R4 are herein defined, said compounds being novel antagonists for melanin-concentrating hormone (MCH), as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising such MCH antagonists as well as methods of using them to treat obesity, metabolic disorders, eating disorders such as hyperphagia, and diabetes.
priorityDate 2003-08-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 485.