http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-2526082-C

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-02
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4196
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filingDate 2004-05-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2012-07-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_308aff6335e8ad989178a0952794dbe5
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_905c12525a68701fbf050286bdb6666a
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3d2122703f86198e111e0fca80cfd259
publicationDate 2012-07-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2526082-C
titleOfInvention Triazole-derivatives as factor xa inhibitors
abstract The present invention relates to compounds of the formulae (I) and (II), in which RO; R1; R3; Q; J1; J2; J3; J4; J5; V; G and M have the meanings indicated in the claims. The compounds of the formulae (I) and (II) are valuable pharmacologically active compounds. They exhibit a strong antithrombotic effect and are suitable, for example, for the therapy and prophylaxis of cardiovascular disorders like thromboembolic diseases or restenoses. They are reversible inhibitors of the blood clotting enzymes factor Xa (FXa) and/or factor VIIa (FVIIa), and can in general be applied in conditions in which an undesired activity of factor Xa and/or factor VIIa is present or for the cure or prevention of which an inhibition of factor Xa and/or factor VIIa is intended. The invention furthermore relates to processes for the preparation of compounds of the formulae (I) and (II), their use, in particular as active ingredients in pharmaceuticals, and pharmaceutical preparations comprising them.
priorityDate 2003-05-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21465112
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559278
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393637
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420251766
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411471142
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450859897
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11150146
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456144919
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408977279
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9262
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450237675
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID640539
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419578441
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5461042
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID536683
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12429372
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419546884
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409782579
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID94395
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450461534
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426247724
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19799
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419576306
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12657
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59149
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9266
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406908050
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67519
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457802510
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424859681
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409783661
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415854255
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID231360
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457798390
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419578766
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166734
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419567129
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415739720

Total number of triples: 341.