http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-2525886-C

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D295-185
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C311-32
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filingDate 2004-05-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-01-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3f88ada3fa80892bb1283f911eb6f23c
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_21b3565f74fb714ef74a1e8dd33e32cf
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fe7594c588c239a3be4fbd7b9a31244b
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publicationDate 2013-01-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2525886-C
titleOfInvention N-sulphonylated amino acid derivatives and their use as matriptase inhibitors
abstract The present invention relates to N-sulfonylated amino acid derivatives, where an aryl radical is linked via the sulfonyl group N-terminally to the amino acid and a radical which comprises at least one imino group and at least one further basic group which represents an optionally modified amino, amidino or guanidino group is linked C--terminally via the carbonyl group. The invention likewise relates to processes for preparing these compounds and to their use, in particular as inhibitors of matriptase.
priorityDate 2003-05-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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