http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-2496585-C

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-08
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filingDate 2003-09-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2012-05-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8c167f0bc0f3191eddab72c8acf57cc5
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6fc1ff18ff049054e0bc4653753c307d
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9f65cf9fc24a3bb536cf1858b324ae34
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_74dfb0f9458094bfb9bdb2bf6bcb8576
publicationDate 2012-05-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2496585-C
titleOfInvention Novel 1,4-diazabicycloalkane derivatives, their preparation and use
abstract This invention relates to novel 1,4-diazabicycloalkane derivatives of formula (I): any of its enantiomers or any mixture of its enantiomers, or a pharmaceutically-acceptable addition salt thereof, or an N-oxide thereof, and their use in the manufacture of pharmaceutical compositions. The compounds of the invention are found to be cholinergic ligands at the nicotinic acetylcholine receptors and modulators of the monoamine receptors and transporters. Due to their pharmacological profile the compounds of the invention may be useful for the treatment of diseases or disorders as diverse as those related to the cholinergic system of the central nervous system (CNS), the peripheral nervous system (PNS), diseases or disorders related to smooth muscle contraction, endocrine diseases or disorders, diseases or disorders related to neuro-degeneration, diseases or disorders related to inflammation, pain, and withdrawal symptoms caused by the termination of abuse of chemical substances.
priorityDate 2002-09-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 411.