http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-2451798-A1

Outgoing Links

Predicate Object
assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_bcb902180030429383f2a70cd2354eaf
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/G01N2500-04
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/G01N33-942
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-4545
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-343
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-343
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/G01N33-94
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4545
filingDate 2003-12-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_cf377e56ee32ed34f1e34e6baeea5aed
publicationDate 2005-06-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2451798-A1
titleOfInvention Use of d4 and 5-ht2a antagonists, inverse agonists or partial agonists
abstract The present invention relates to the use of compounds and compositions of compounds having D4 and/or 5-HT2A antagonistic, partial agonistic or inverse agonistic activity for the treatment of the underlying dysregulation of the emotional functionality of mental disorders (i.e. affect instability - hypersensitivity - hyperaesthesia - dissociative phenomena -...). The invention also relates to methods comprising administering to a patient diagnosed as having a neuropsychiatric disorder a pharmaceutical composition containing (i) compounds having D4 antagonistic, partial agonistic or inverse agonistic activity and/or (ii) compounds having 5-HT2A antagonistic, partial agonistic or inverse agonistic, and/or (iii) any known medicinal compound and compositions of said compounds. The combined D4 and 5-HT2A antagonistic, partial agonistic or inverse agonistic effects may reside within the same chemical or biological compound or in two different chemical and/or biological compounds.
priorityDate 2003-12-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

Incoming Links

Predicate Subject
isDiscussedBy http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23573
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3372
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480399
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60835
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2771
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54676228
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID151166
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419493602
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501289
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4748
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480882
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68617
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID123619
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419592003
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3058754
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480562
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID33014
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2726
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5736
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5656
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410111933
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419499849
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119828
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419475708
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID55752
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419494663
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3396
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135398745
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419494789
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419495692
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419494657
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2159
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID125564
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID37825
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID219077
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID184841
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419536136
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419476058
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406917592
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506685
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3559
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5452
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419499092
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419498333
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2662
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419495644
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419499404
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3386
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135515430
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480116
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506816
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507641
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71360
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5090
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID72036
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135398737
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415136092
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9922854
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119607
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID73333
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4830
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID65833
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492896
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60795
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID43815
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507434
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419505781
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419553097
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6918388
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415220896
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507378
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480990
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412892589
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54841
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419533756
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507450
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409050809
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419495697
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID431429
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415868268
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424977963
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415728329
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3033769
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID20055529
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419498766
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6917700
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5666
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507566
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4528
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5073
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419552831
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419497667
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5361192
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71351
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54677470
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID127151
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5566
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410878039
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415718916
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136319
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419533573
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492710
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60785
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507462
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506282
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504025
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425701257
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60149
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507324
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506457
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419499387
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534410
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507599
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60854
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5002
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID133079
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501547
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID39187
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419490957
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507269
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4078
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501145

Total number of triples: 141.