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publicationDate 2008-03-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2429378-C
titleOfInvention Improved process for water soluble azole compounds
abstract An improved process is provided for preparing water-soluble prodrugs of triazole antifungal compounds containing a secondary or tertiary hydroxyl group. More particularly, the improved process is directed toward preparation of water-soluble triazole antifungal compounds having the general formula (I) wherein A is the non-hydroxy portion of a triazole antifungal compound of the type containing a secondary or tertiary hydroxyl group and R and R1 are as defined in the specification.
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