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filingDate 1996-04-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_caf9515b11e4317785aed2b88cdf9356
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publicationDate 1996-10-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CA-2218597-A1
titleOfInvention Cyclobutane derivatives as inhibitors of squalene synthase and protein farnesyltransferase
abstract The present invention provides a compound of formula (I) or (II) or a pharmaceutically acceptable salt thereof, which is useful for inhibiting protein farnesyltransferase and the farnesylation of the oncogene protein Ras or inhibiting de novo squalene production resulting in the inhibition of cholesterol biosynthesis, processes for the preparation of the compounds of the invention in addition to intermediates useful in these processes, a pharmaceutical composition, and to methods of using such compounds.
priorityDate 1995-04-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 422.