http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-2187429-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_620ecb9324409347c27e96b6071503ee |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-14 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-14 |
| filingDate | 1995-04-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c344d8e3fc0800667200821b40cbff83 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_96b21155d64298e17085fd491ee5062a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c0b572d50017076e67225e02d5fbbc84 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9b9dbe8a94e6f220c434e2bb4705bef5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5e578fdfa030c86cf5dac2ae51a3c984 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bb7a62a44255031afd7b551d92f78bb1 |
| publicationDate | 1995-11-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CA-2187429-A1 |
| titleOfInvention | N-(3-pyrrolidinyl)benzamide derivative |
| abstract | An N-(3-pyrrolidinyl)benzamide derivative represented by general formula (I) or a pharmaceutically acceptable salt thereof and a medicine containing the same, having a potent and selective antagonism against dopamine D3 and/or D4 receptors and useful as a psychotropic agent, schizophrenia remedy, and so forth. In said formula, R1 represents hydrogen, lower alkyl, aralkyl, or three-to eight-membered cycloalkyl or cycloalkyl-lower alkyl; R2 represents four-to sixteen-membered bi- or tricyclic bridged hydrocarbon group; R3 represents lower alkoxy, amino, or mono- or di(lower alkyl)amino; R4 represents hydrogen, halogen, optionally hydroxylated lower alkyl, lower alkoxy, cyano, nitro, amino, mono- or di(lower alkyl)amino, acyl or -S(O)m-R5; R5 represents lower alkyl, amino or mono- or di(lower alkyl)amino; m represents 0, 1 or 2; X represents a bond, -O-, -S(O)n-, -NH- or -CONH-; and n represents 0, 1 or 2; provided when R1 represents cycloalkyl, the case where X represents -CONH-, R3 represents lower alkoxy and R4 represents halogen is excepted. |
| priorityDate | 1994-04-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 282.