http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-2103242-C
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-55 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D519-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K33-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D235-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P37-08 |
| filingDate | 1992-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2002-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_702ee87d99ee3a476df0c10771fe228b http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f98c21b0bf99296f07223544103961ed http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_31483d9ffb257ec06c4056680b5cc866 |
| publicationDate | 2002-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CA-2103242-C |
| titleOfInvention | Imidazo[2,1-b][3]benzazepine derivatives, compositions and method of use |
| abstract | The present invention is concerned with novel imidazo[2,1-b][3]benzazepines of formula (I), the pharmaceutically accept-able addition salts and stereochemically isomeric forms thereof, wherein each of the dotted lines independently represents an op-tional bond; R1 represents hydrogen, halo, C1-4alkyl or C1-4alkyloxy; R2 represents hydrogen, halo, C1-4alkyl or C1-4alky-loxy; R3 represents hydrogen, C1-4alkyl, ethenyl substituted with hydroxycarbonyl or C1-4alkyloxycarbonyl, C1-4alkyl substi-tuted with hydroxycarbonyl or C1-4alkyloxycarbonyl, hydroxyC1-4alkyl, formyl or hydroxycarbonyl; R4 represents hydrog-en, C1-4alkyl, hydroxyC1-4alkyl, phenyl or halo; R5 represents hydrogen, C1-4alkyl or halo; L represents hydrogen; C1-6al-kyl; C1-6alkyl substituted with one substituent selected from the group consisting of hydroxy, halo, C1-4alkyloxy, hydroxy-carbonyl, C1-4alkyloxycarbonyl, C1-4alkyloxycarbonyl-C1-4alkyloxy, hydroxycarbonylC1-4alkyloxy, C1-4alkyloxycarbony-lamino, C1-4alkylaminocarbonyl, C1-4alkylaminocarbonylamino, C1-4alkylaminothiocarbonylamino, aryl, aryloxy and aryl-carbonyl; C1-6alkyl substituted with both hydroxy and aryloxy; C3-6alkenyl; C3-6alkenyl substituted with aryl; or, L repres-ents a radical of formula -Alk-Y-Het1 (a-1), -Alk-NH-CO-Het2 (a-2) or -Alk-Het3 (a-3); provided that 6,11-dihydro-11-(4-piperidinylidene)-5H-imidazo[2,1-b][3]benzazepine is excluded, which are useful antiallergic compounds. Compositions comprising said compounds, methods of using and processes for preparing the same. |
| priorityDate | 1991-06-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 298.