http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-1272213-A
Outgoing Links
Predicate | Object |
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assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_5c24684033fba97d1ad845ce453a57e3 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C255-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D263-14 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C217-32 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C217-30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C67-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B31-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D263-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C213-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B55-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B53-00 |
filingDate | 1983-08-03-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate | 1990-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7fd330d5cd458152d2de6d39dc1c60ec http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_539ac6f5b176a88ac63d733dfabdc1a0 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_447ac5b97c8dc69b7d7a80a75a073335 |
publicationDate | 1990-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | CA-1272213-A |
titleOfInvention | Process for inverting the configuration of optically active compounds, and optically active intermediates produced in this process |
abstract | ABSTRACT OF THE INVENTION The invention relates to a process for inverting the configuration at the optically active carbon atom (*) in compounds of the formula I (I) in which A denotes a carbocyclic or heterocyclic aromatic radical and R denotes an aliphatic, cycloaliphatic or araliphatic hydrocarbon radical, by formylation, treating the resulting compounds with a strong acid or an acid halide and cleaving the oxazolinium derivatives thus obtained, by acid or alkaline hydrolysis, if appropriate via the stage of the N-formyl compound, and to oxazolinium derivatives of the formula III (III) in which A and R have the meanings defined above and in which X? represents the anion of a strong acid or of a halogen atom and formed as intermediate products. Compounds of the formula IV (IV) in which A and R have the meanings defined above, possessing the same structure as the starting material I but having an opposite configuration at the carbon atom (*), can be used as .beta.-blocking agents. |
priorityDate | 1982-08-04-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 81.