http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-1260475-A
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_da54f7ebbd2d9d8a82f92aca4d1b4e48 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-4015 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-6561 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F9-6561 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F9-40 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-44 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-675 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-435 |
| filingDate | 1983-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 1989-09-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_72a363be0bcae8a9c1cb7123986d5180 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_550b6f992f5e8071e4bb0df2de03d502 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_517131970211294fc11ee377354b53e8 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_545fa26f906cde02de109c93000539e9 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7f85180101001463316342cf1b51693b http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_552bdf8d20301df1fba69c71f019356e |
| publicationDate | 1989-09-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CA-1260475-A |
| titleOfInvention | .beta.-CARBOLINES, PROCESS FOR THEIR PRODUCTION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM |
| abstract | ABSTRACT OF THE DISCLOSURE A .beta.-carboline of the formula wherein R3 is halogen; ORI, wherein RI is H, C1-5 alkyl, C3-7-cycloalkyl, C7-10-aralkyl or C6-10-aryl; NRIIRIII, wherein RII is H, C1-5alkyl, C3-7-cycloalkyl. C7-10-aralkyl or C6-10 aryl and RIII is C1-5 alkyl. C1-3-alkanoyl, C1-6 alkoxycarbonyl, carbamoyl, or RII and RIII together with the connecting N-atom are pyrrolyl or piperidino; SOnRI, wherein n is 0, 1 or 2 and RI is as defined above; PO3RIVRV, wherein RIV each independently is H, C1-5-alkyl, C3-7-cycloalkyl, C7-10-aralkyl or C6-10 aryl; or C3-7-cycloalkyl, C8-12-aralkenyl, or C6-10-aryl, each of whose alkyl portion may be substituted by 1 to 3 of halogen, OR,INRIIRIII, SOnRI, COORI, CONRIIRIII, CSNRIIRIII, PO3RIVRV, CORI or CN, wherein RI, RII, RIII, RIV, RV and n are as defined above; R4 is H, C1-5 alkyl, C1-5 alkoxy-C1-5-alkyl, CORVI or CSRVII, wherein RVI is H, C1-5-alkyl, C3-7-cycloalkyl, C7-10-aralkyl, OH, O-C1-5-alkyl, O-C3-7-cycloalkyl, O-C7-10-aralkyl or NRIIRII, wherein RII is as defined above and the RII's can be the same or different or both RII's together with the N are pyrrolyl or piperidino and wherein RVII is H, C1-5 alkyl, C3-7-cycloalkyl or C7-10-aralkyl; R5-R8 each independently is H, halogen NO2, ORI, NRIIRIII, PO3RIVRV, SO2NRIRV, COORI, CONRIIRIII, CSNRIIRIII and CORI wherein RI-V are as defined above and at most two of R5-R8 can be non-H; and R9 is H, C1-5 alkyl, C1-3-alkanoyl, carbamoyl, C1-6-alkoxycarbonyl, or SO2RVIII wherein RVIII is methyl or p-tolyl are valuable pharmaceutical products with long lasting action on the central nervous system. |
| priorityDate | 1982-10-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 179.