http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-1167845-A
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_a7f82940e47ba7a1188f8e2ffca55e0f |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D213-73 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-435 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P1-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D213-73 |
| filingDate | 1981-01-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 1984-05-22-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_868f66a4da8d675c6e137e0af07faa1c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4ccc3b64c1baa38cc760f9dcbd52552a |
| publicationDate | 1984-05-22-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | CA-1167845-A |
| titleOfInvention | Imidazo¬1,2-a|pyridines, processes for their preparation and pharmaceutical compositions containing them |
| abstract | A B S T R A C T The invention relates to imidazo[1,2-a] pyridines of the general formula wherein R2 represents hydrogen, lower alkyl, trifluoromethyl, B-CF3; B-Ar, Ar, B-halogen, BOR8, B-SO(n)-loweralkyl, BO?-R1, ; R3 represents loweralkyl, BCN, BOR8, BO?-R1, B-NO2, B-halogen or, provided R2 is not hydrogen, hydrogen; X is hydrogen, loweralkyl, halogen, hydroxy, trifluoro-methyl or loweralkoxy; Z represents O, S, SO, SO2, NR6 or a single bond between the group T-Ar and position 8 of the imidazo [1,2-a]pyridine nucleus; T represents a single bond between Z and Ar or a branched or straight alkylene group having 1 to 12 carbon atoms with no more than 5 binding carbon atoms between Z and Ar; and Ar represents phenyl, pyridyl, thienyl, furanyl, imidazolyl or X'-, Y'- and/or Z'-substituted phenyl wherein each of X', Y' and Z' independently is hydrogen, halogen, loweralkyl, loweralkoxy, CN, CF3, OH, NO2, or SO(m)-R1, with m being zero, one or two, whereby m represents two when R1 represents whereby in the above definitions B is a straight or branched chain lower alkylene group; n represents zero, one or two; R4 and R5 eacn independently represent hydrogen, loweralkyl, loweralkyl, loweralkoxyloweralkyl trifluoromethyllower-alkyl, Ar-loweralkyl, Ar, or, when taken together with the nitrogen to which they are attached, form a 4- to 6-membered cyclic amino- or a morpholino-group; R1 represents Ar, loweralkyl, or Ar-lower-alkyl; R6 represents hydrogen, C1- to C12-alkyl, aryl-or an aralkyl group having up to 12 carbon atoms. R7 represents hydrogen or loweralkyl and R8 represents hydrogen, loweralkyl,loweralkoxyloweralkyl, trifluoro-methylloweralkyl, Ar-loweralkyl or Ar. |
| priorityDate | 1980-01-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
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