http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CA-1153366-A
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_0e77f06144be4708a6ae75bd9fee56a4 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J43-003 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-58 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07J43-00 |
filingDate | 1980-12-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate | 1983-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3bea2780e906b35bd21dfa76b2e7e65a |
publicationDate | 1983-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | CA-1153366-A |
titleOfInvention | BIS- AND MONO-QUATERNARY AMMONIUM DERIVATIVES OF 2.beta., 16.beta.-DIPIPERIDINO-5.alpha.-ANDROSTANES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS |
abstract | ABSTRACT The invention relates to novel bisquaternary ammonium derivatives of 2.beta.,16.beta.-dipiperidino-5.alpha.-androstanes having the formula: .2X-wherein ; R2 = CH3, C2H5 or CH2CH=CH2; R3 = CH3, C2H5 or CH2CH=CH2, with the proviso that R2 and R3 are not CH3 simultaneously; R4 = O or H(.beta.OR5), wherein R5 = H or aliphatic carbacyl (1-6 C); and X = a halogen atom, to processes for their preparation and to pharmaceutical preparations. The invention also relates to novel 16-monoquaternary analogs as intermediates. The compounds possess neuromuscular blocking activity. |
priorityDate | 1979-12-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 62.