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publicationDate 2021-05-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber BR-PI0718436-B8
titleOfInvention bradykinin b1 receptor antagonist compounds derived from phenylsulfamoylbenzamide, process for preparing the same, their use and pharmaceutical composition
abstract new benzamide derivatives as bradykinin antagonists. the present invention relates to novel phenylsulfamoylbenzamide derivatives of formula (I), wherein r1-r5 are as defined in the claims, and optical antipodes or racemates and/or salts and/or hydrates and/or solvates thereof, which are antagonists selective bradykinin b1, processes for producing these compounds, pharmaceutical compositions containing them, and their uses in the therapy or prevention of painful and inflammatory conditions.
priorityDate 2006-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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