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filingDate 2001-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bb70df56b2e4e612632c6cd6ff5da823
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publicationDate 2018-04-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber BR-PI0113146-B1
titleOfInvention "PROLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION UNDERSTANDING THEM".
abstract "proline derivatives and their use as drugs". The present invention relates to the provision of compounds having therapeutic effects due to an inhibitory action of dpp-iv, and satisfactory as pharmaceuticals. The present inventors have found that derivatives having a substituent introduced at the proline y position represented by formula (1) wherein each symbol is defined in the specification, have potent dpp-iv inhibitory activity, and have completed the present invention by increasing the stability.
priorityDate 2000-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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