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filingDate 2019-12-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d03bb81964bca5e812afeaf752e8ea6a
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eb99b60039c6a7ebe9fc64c060b67fa1
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publicationDate 2021-08-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber BR-112021010842-A2
titleOfInvention 2-Oxoquinazoline Derivatives as Methionine Adenosyltransferase 2a Inhibitors
abstract The present invention relates to certain 2-oxoquinazoline derivatives of formula (ia): (ia) which are inhibitors of methionine adenosyltransferase 2a (mat2a). pharmaceutical compositions comprising such compounds and methods of treating diseases treatable through inhibition of mat2a, such as cancer, including cancers characterized by reduced or no activity of methylthioadenosine phosphorylase (mtap) are also described.
priorityDate 2018-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1213.