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publicationDate 2022-08-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber BR-112017004209-B1
titleOfInvention COMPOUNDS DERIVED FROM TETRAHYDRONAPHTHALENE, PHARMACEUTICAL COMPOSITION AND USE THEREOF TO INHIBITS MCL-1 PROTEIN
abstract TETRAHYDRONAPHTHALENE DERIVATIVES WHICH INHIBIT MCL-1 PROTEIN. Presented herein are myeloid cell leukemia protein 1 (Mcl-1) inhibitors, methods for their preparation, related pharmaceutical compositions, and methods of using the same. For example, compounds of Formula I, (I) and pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the compounds are disclosed herein. The compounds and compositions presented herein can be used, for example, in the treatment of diseases or conditions, such as cancer.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25074887
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5790
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118910331
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25074470
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID439888
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD4A9L7
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135410875
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581812
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12291149
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118910333
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14055602
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2064
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71308305
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118903436
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53232
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95KP3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13781592
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426079013
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422951417
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419500673
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5329102
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3305
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID15965
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118903753
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152774259
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407064580
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373954
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118910355
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407275646
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID374569
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9824723
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414803645
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3276
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID45083885

Total number of triples: 1284.