http://rdf.ncbi.nlm.nih.gov/pubchem/patent/BR-112015014839-B1

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filingDate 2013-12-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5ce1abfd899e46d9c34db0d894fdae3e
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publicationDate 2022-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber BR-112015014839-B1
titleOfInvention CRYSTALLINE FORM OF THE COMPOUND USED AS A MINERALOCORTICOID RECEPTOR ANTAGONIST, ITS USES, ITS PREPARATION PROCESS AND PHARMACEUTICAL COMPOSITION
abstract CRYSTALLINE FORM OF THE COMPOUND USED AS A MINERALOCORTICOID RECEPTOR ANTAGONIST AND METHOD FOR THEIR PREPARATION. The present invention pertains to the technical field of medicaments, and relates to a crystalline form of a compound used as a mineralocorticoid receptor antagonist and a method for its preparation, and in particular, a method for the preparation of a compound 2-chloro-4-[(3S,3aR)-3-cyclopentyl-7-(4-hydroxypiperidine-1-carbonyl)-3,3a,4,5-tetrahydro-2H-pyrazolo[3,4-f]quinoline -2-yl]benzonitrile of formula (I), a crystalline form thereof, a method of preparation for the crystalline form, and the use of the crystalline form in the preparation of medicaments for the treatment and/or prevention of kidney damage or cardiovascular diseases.
priorityDate 2012-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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