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filingDate 2010-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2021-06-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber BR-112012021911-B1
titleOfInvention process for the production of pyripyropene derivatives
abstract process for the production of pyripyropene derivatives. a process for the production of pyripyropene derivatives having acyloxy at position 1 and 11 and hydroxyl at position 7 is presented. The process consists of selective acylation of hydroxyl at position 1 and at position 11 of a compound represented by formula b1 through one or three steps, with an acylating agent in the presence or absence of a base.
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