| abstract |
"BENZIMIDAZOLE COMPOUNDS AND ITS USE AS STROGEN AGONISTS / ANTAGONISTS". The present invention relates to compounds of formula (I) or a pharmaceutically acceptable salt thereof, wherein at least one of R3 and R3 is a group of formula (II) wherein R7 , R48. R 9, R 10 and R 11 are independently from each other hydrogen; hydroxy; (C 1-1 -C 6) alkyl; (C1-6 -C6) alkoxy; or halogen; R9 is hydroxy; (C1-6 -C6) alkoxy; (C 1 -C 6) alkoxycarbonyloxy; (C 3 -C 8) cycloalkoxy; (C 4-4 -C 8) cycloalkenyloxy; or (C 6 -C 12) aryloxy; which are useful as estrogen agonists and / or antagonists and their pharmaceutical uses. |