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publicationDate 2009-12-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber BG-110141-A
titleOfInvention GALANTAMINE DERIVATIVES, METHODS FOR THEIR PREPARATION AND USE
abstract The invention relates to novel compounds which are galanthamine derivatives, to processes for their preparation and to their use for the prophylaxis and / or treatment of neurodegenerative diseases, including senile dementia and Alzheimer's disease. The novel galanthamine derivatives according to the invention combine two effects: inhibition of acetylcholinesterase and butyrylcholinesterase activity due to the galanthamine molecule and inhibition of gamma-secreting activity inherent in the peptide fragment.
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