http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AU-2017339786-A1

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publicationDate 2019-05-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2017339786-A1
titleOfInvention Bryostatin compounds and methods of preparing the same
abstract Methods for preparing a variety of bryostatin compounds are provided. The subject methods provide for preparation of bryostatin 1 in multi-gram quantities in a low and unprecedented number of convergent synthetic steps from commercially available materials. The subject methods are scalable with low estimated material costs and can provide enough material to meet clinical needs. Also provided are a variety of bryostatin analog compounds, and prodrug forms thereof, which are synthetically accessible via the subject methods and pharmaceutical compositions including the same.
priorityDate 2016-10-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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