http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AU-2017202446-B2

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filingDate 2017-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_cc9ddbbd953855b69c577d9db237a22d
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publicationDate 2019-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2017202446-B2
titleOfInvention Process for manufacturing pyrimidine sulfamide derivatives
abstract - 51 The invention relates to a process for manufacturing the compound of formula I 0 \1 r110 R O O Br Br 5 wherein R is H, (C-C6 )alkyl or benzyl. or a salt thereof, said process comprising the reaction of the compound of formula 1-1 Br NN O Br I-1 wherein X is Br, Cl or F, or a salt thereof, with the compound of formula 1-2 o o 1-2 wherein R is H, (CI-C6 )alkyl or benzyl, or a salt thereof, in the presence of a base, and, when X is Br or Cl, in the presence of tetra-n-butyl ammonium fluoride hydrate or cesium 10 fluoride. The invention further relates to the compound of formula I-I and uses thereof.
priorityDate 2014-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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