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filingDate 2016-06-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-01-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_641428d8c6760f2015807c594d9a0b93
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publicationDate 2020-01-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2016279518-B2
titleOfInvention Imidazodiazepine compound
abstract [Problem] To provide a compound useful as a dopamine D1 receptor positive allosteric modulator (D1 PAM). [Solution] The present inventors have studied on compounds each of which has a positive allosteric modulating activity (a PAM activity) on a dopamine D1 receptor and can be used as an active ingredient for a prophylactic or therapeutic pharmaceutical composition for cognitive dysfunction, schizophrenia negative symptoms, CIAS, Parkinson's disease, Alzheimer's disease, Huntington's disease, depression, ADHD, drug dependence and the like. As a result, it is confirmed that an imidazodiazepine compound according to the present invention has a PAM activity on a dopamine D1 receptor, and the present invention has been accomplished. The imidazodiazepine compound according to the present invention has a PAM activity on a dopamine D1 receptor and is expected to be used as a prophylactic and/or therapeutic agent for cognitive dysfunction, schizophrenia negative symptoms, CIAS, Parkinson's disease, Alzheimer's disease, Huntington's disease, depression, ADHD, drug dependence and the like.
priorityDate 2015-06-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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