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publicationDate 2016-11-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2016244296-A1
titleOfInvention Process for Making Modulators of Cystic Fibrosis Transmembrane Conductance Regulator
abstract The invention provides a process for the preparation of a compound of Formula 1, N H (Rx-X H R2 Formula 1 comprising coupling a carboxylic acid of Formula 2 (Rx-X OH Formula 2 with an aniline of Formula 3 Formula 3 in the presence of a coupling agent.
priorityDate 2009-03-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 545.