http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AU-2012324032-B2

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titleOfInvention Gel compositions
abstract (12) INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (10) International Publication Number (43) International Publication Date W O 2013/088375 Al 20 June 2013 (20.06.2013) WI PO I P CT (51) International Patent Classification: (81) Designated States (unless otherwise indicated, for every A61K 9/06 (2006.01) A61K 9/00 (2006.01) kind of national protection available): AE, AG, AL, AM, A61K31/22 (2006.01) A61K 47/24 (2006.01) AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, ) .a BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, (21) International Application Number: DO, DZ, EC, EE, EG, ES, Fl, GB, GD, GE, GH, GM, GT, PCT/IB2012/057250 HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, (22) International Filing Date: KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, 12 December 2012 (12.12.2012) ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, (25) Filing Language: English RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, (26) Publication Language: English TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW. (30) Priority Data: 61/569,643 12 December 2011 (12.12.2011) US (84) Designated States (unless otherwise indicated, for every kind of regional protection available): ARIPO (BW, GH, (71) Applicant: LEO LABORATORIES LIMITED [IE/IE]; GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, 285 Cashel Road, Crumlin, Dublin, 2 (IE). UG, ZM, ZW), Eurasian (AM, AZ, BY, KG, KZ, RU, TJ, (72) Inventors: Arvidsson, Per Ola; LEO Pharma A/S, Indus- TM), European (AL, AT, BE, BG, CH, CY, CZ, DE, DK, triparken 55, DK-2750 Ballerup (DK). Farkas, Edit; LEO EE, ES, Fl, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, Pharma A/S, Industriparken 55, DK-2750 Ballerup (DK). MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, Petersson, Karsten; LEO Pharma A/S, Industriparken 55, TR), OAPI (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, DK-2750 Ballerup (DK). Hoy, Gert; LEO Pharma A/S, In- ML, MR, NE, SN, TD, TG). dustriparken 55, DK-2750 Ballerup (DK). Published: (74) Agents: MARSHALL, Cameron John et al.; Carpmaels - with international search report (Art. 21(3)) & Ransford, One Southampton Row, London WC 1 B 5HA (GB). (54) Title: A TOPICAL COMPOSITION COMPRISING AN INGENOL DERIVATIVE AND AN OILY SOLVENT (57) Abstract: A substantially anhydrous topical composition comprises a homogenous mixture of (a) a therapeutically effective amount of an ingenol derivative in dissolved form; (b) an oily solvent for the ingenol derivative, (c) an acidic compound, and (d) op tionally a pharmaceutically acceptable non-solvent lipid carrier.
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